TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of human Mcl-1 assessed as inhibition constant by DELFIA displacement assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of human Mcl-1 assessed as inhibition constant by DELFIA displacement assayMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 7(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataKi: 185nMAssay Description:Binding affinity to N-terminal His-tagged wild type ML-IAP BIR domain (63 to 179 residues) (unknown origin) expressed in Escherichia coli BL21 assess...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Displacement of AVPIAQKSEK-biotin from cIAP1 BIR3 (unknown origin) after 1 hr by DELFIAMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of EPHA2 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of EPHA2 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Inhibition of EPHA2 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 7(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Antagonist activity at N-terminal His-tagged wild type ML-IAP BIR domain (63 to 179 residues) (unknown origin) expressed in Escherichia coli BL21 usi...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 9.30nMAssay Description:Inhibition of EPHA2 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of AVPIAQKSEK-biotin from cIAP1 BIR3 (unknown origin) after 1 hr by DELFIAMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Displacement of AVPIAQKSEK-biotin from N-terminal His-tagged human recombinant XIAP BIR3 (253 to 347 residues) expressed in Escherichia coli BL21(DE3...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of EPHA2 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 7(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at N-terminal His-tagged wild type ML-IAP BIR domain (63 to 179 residues)(unknown origin) expressed in Escherichia coli BL21 usin...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Displacement of AVPIAQKSEK-biotin from cIAP2 BIR3 (unknown origin) after 1 hr by DELFIAMore data for this Ligand-Target Pair
Affinity DataIC50: 13.9nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of EPHA2 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 7(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Antagonist activity at N-terminal His-tagged wild type ML-IAP BIR domain (63 to 179 residues)(unknown origin) expressed in Escherichia coli BL21 usin...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Displacement of AVPIAQKSEK-biotin from cIAP2 BIR3 (unknown origin) after 1 hr by DELFIAMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Antagonist activity at N-terminal His-tagged cIAP1-BIR3 domain (unknown origin) expressed in Escherichia coli BL21 using AVPIAQKSEK-biotinylated pept...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonist activity at N-terminal His-tagged cIAP2-BIR3 domain (unknown origin) expressed in Escherichia coli BL21 using AVPIAQKSEK-biotinylated pept...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of AVPIAQKSEK-biotin from N-terminal His-tagged human recombinant XIAP BIR3 (253 to 347 residues) expressed in Escherichia coli BL21(DE3...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of AVPIAQKSEK-biotin from cIAP1 BIR3 (unknown origin) after 1 hr by DELFIAMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonist activity at N-terminal His-tagged cIAP2-BIR3 domain (unknown origin) expressed in Escherichia coli BL21 using AVPIAQKSEK-biotinylated pept...More data for this Ligand-Target Pair
TargetBcl-2-related protein A1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 7(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at N-terminal His-tagged wild type ML-IAP BIR domain (63 to 179 residues) (unknown origin) expressed in Escherichia coli BL21 usi...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Displacement of AVPIAQKSEK-biotin from XIAP BIR3 Lys322A mutant (unknown origin) after 1 hr by DELFIAMore data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of EPHA2 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Antagonist activity at N-terminal His-tagged cIAP1-BIR3 domain (unknown origin) expressed in Escherichia coli BL21 using AVPIAQKSEK-biotinylated pept...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Displacement of AVPIAQKSEK-biotin from cIAP1 BIR3 (unknown origin) after 1 hr by DELFIAMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Displacement of AVPIAQKSEK-biotin from N-terminal His-tagged human recombinant XIAP BIR3 (253 to 347 residues) expressed in Escherichia coli BL21(DE3...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Displacement of AVPIAQKSEK-biotin from cIAP1 BIR3 (unknown origin) after 1 hr by DELFIAMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair